Titre:
  • A novel chalcone derivative which acts as a microtubule depolymerising agent and an inhibitor of P-gp and BCRP in in-vitro and in-vivo glioblastoma models.
Auteur:Boumendjel, Ahcène; McLeer-Florin, Anne; Champelovier, Pierre; Allegro, Diane; Muhammad, Dima; Souard, Florence; Derouazi, Madiha; Peyrot, Vincent; Toussaint, Bertrand; Boutonnat, Jean
Informations sur la publication:BMC cancer, 9, page (242)
Statut de publication:Publié, 2009-07
Sujet CREF:Sciences bio-médicales et agricoles
MeSH keywords:ATP Binding Cassette Transporter, Subfamily B, Member 1 -- antagonists & inhibitors -- metabolism
Animals
Antineoplastic Agents -- pharmacology
Apoptosis
Blood-Brain Barrier
Brain Neoplasms -- metabolism
Cell Line, Tumor
Chalcone -- analogs & derivatives
Chalcones -- pharmacology
Glioblastoma -- metabolism
Humans
Mice
Mice, Inbred C57BL
Microtubules -- metabolism
Proto-Oncogene Proteins c-bcr -- antagonists & inhibitors -- metabolism
Rats
Langue:Anglais
Identificateurs:urn:issn:1471-2407
info:doi/10.1186/1471-2407-9-242
info:pii/1471-2407-9-242
info:pmid/19619277
PMC2717121