par Gigot, Daniel 
;Penninckx, Michel
Référence Journal of pharmaceutical sciences, 73, 2, page (275-277)
Publication Publié, 1984-02
;Penninckx, Michel Référence Journal of pharmaceutical sciences, 73, 2, page (275-277)
Publication Publié, 1984-02
Article révisé par les pairs
| Résumé : | Two peptide forms of the antitumor transition state analogue N-phosphonoacetyl-L-aspartic acid (N2-phosphonoacetyl-N4-glycylglycinamidoethyl-L-asparagine and N1-glycylglycinamidoethyl-N2-phosphonoacetyl-L-isoasparagine ) have been synthesized to obtain potential medicinal agents useful as prodrugs or in a lysosomotropic carrier approach. The bridging unit, ethylenediamine, used for synthetic purposes might be of general interest. |
