Titre:
  • Activation of guanosine 5'-[gamma-(35)S]thio-triphosphate binding through M(1) muscarinic receptors in transfected Chinese Hamster ovary cell membranes: 2. Testing the "two-states" model of receptor activation.
Auteur:Waelbroeck, Magali
Informations sur la publication:Molecular pharmacology, 59, 4, page (886-893)
Statut de publication:Publié, 2001-04
Sujet CREF:Sciences bio-médicales et agricoles
MeSH keywords:Animals
Binding, Competitive -- drug effects
CHO Cells
Cell Membrane -- metabolism
Cricetinae
Dose-Response Relationship, Drug
GTP-Binding Protein alpha Subunits, Gi-Go -- antagonists & inhibitors
Guanosine 5'-O-(3-Thiotriphosphate) -- metabolism
Guanosine 5'-O-(3-Thiotriphosphate) -- pharmacokinetics
Guanosine Diphosphate -- metabolism
Guanosine Triphosphate -- metabolism
Heterotrimeric GTP-Binding Proteins -- antagonists & inhibitors
Models, Biological
Muscarinic Agonists -- metabolism
Muscarinic Agonists -- pharmacology
Pertussis Toxin
Receptor, Muscarinic M1
Receptors, Muscarinic -- genetics
Receptors, Muscarinic -- metabolism
Reproducibility of Results
Sulfur Radioisotopes
Transfection
Virulence Factors, Bordetella -- pharmacology
Note générale:Journal Article
Research Support, Non-U.S. Gov't
Langue:Anglais
Identificateurs:urn:issn:0026-895X
info:pmid/11259634