Titre:
  • Substitution of conserved glycine residue by alanine in natural and synthetic neuropeptide ligands causes partial agonism at the stomoxytachykinin receptor.
Auteur:Poels, Jeroen; Van Loy, Tom; Franssens, Vanessa; Detheux, Michel; Nachman, Ronald J; Oonk, Hendrica B; Akerman, Karl E; Vassart, Gilbert; Parmentier, Marc; De Loof, Arnold; Torfs, Herbert; Broeck, Jozef Vanden
Informations sur la publication:Journal of neurochemistry, 90, 2, page (472-478)
Statut de publication:Publié, 2004-07
Sujet CREF:Sciences bio-médicales et agricoles
Mots-clés:G protein-coupled receptor
Insect
Neuropeptide
Partial agonism
Tachykinin
MeSH keywords:Aequorin -- genetics
Aequorin -- metabolism
Alanine
Amino Acid Sequence
Amino Acid Substitution -- genetics
Amino Acid Substitution -- physiology
Animals
Apoproteins -- genetics
Apoproteins -- metabolism
Biological Assay
Calcium -- metabolism
Cell Line
Conserved Sequence
Cyclic AMP -- metabolism
Dose-Response Relationship, Drug
Drosophila melanogaster
Glycine
Grasshoppers
Insect Proteins -- genetics
Insect Proteins -- metabolism
Insect Proteins -- pharmacology
Ligands
Luminescent Measurements
Molecular Sequence Data
Muscidae
Neuropeptides -- genetics
Neuropeptides -- metabolism
Neuropeptides -- pharmacology
Receptors, Tachykinin -- agonists
Receptors, Tachykinin -- genetics
Receptors, Tachykinin -- metabolism
Recombinant Proteins -- genetics
Recombinant Proteins -- metabolism
Sequence Homology, Amino Acid
Structure-Activity Relationship
Tachykinins -- genetics
Tachykinins -- metabolism
Tachykinins -- pharmacology
Transgenes
Note générale:Journal Article
Research Support, Non-U.S. Gov't
FLWIN
Langue:Anglais
Identificateurs:urn:issn:0022-3042
info:doi/10.1111/j.1471-4159.2004.02506.x
info:pii/JNC2506
info:scp/3142666081
info:pmid/15228603