Titre:
  • New 5-Aryl-1H-imidazoles display in vitro antitumor activity against apoptosis-resistant cancer models, including melanomas, through mitochondrial targeting.
Auteur:Mathieu, Véronique; Van Den Berge, Emilie; Ceusters, Justine; Konopka, Tomasz; Cops, Antonin; Bruyère, Céline; Pirker, Christine; Berger, Walter; Trieu-Van, Tran; Serteyn, Didier; Kiss, Robert; Robiette, Raphael
Informations sur la publication:Journal of medicinal chemistry, 56, 17, page (6626-6637)
Statut de publication:Publié, 2013-09
Sujet CREF:Sciences bio-médicales et agricoles
MeSH keywords:Antineoplastic Agents -- pharmacology
Apoptosis -- drug effects
Cell Line, Tumor
Drug Screening Assays, Antitumor
Humans
Imidazoles -- pharmacology
Melanoma -- pathology
Mitochondria -- drug effects
Models, Biological
Neoplasms -- pathology
Transcriptome
Note générale:Journal Article
Research Support, Non-U.S. Gov't
SCOPUS: ar.j
Langue:Anglais
Identificateurs:urn:issn:0022-2623
info:doi/10.1021/jm400287v
info:scp/84884276750
info:pmid/23845202