Titre:
  • Hydroxylated analogues of ATP-sensitive potassium channel openers belonging to the group of 6- and/or 7-substituted 3-isopropylamino-4H-1,2,4-benzothiadiazine 1,1-dioxides: toward an improvement in sulfonylurea receptor 1 selectivity and metabolism stability.
Auteur:de Tullio, Pascal; Servais, Anne-Catherine; Fillet, Marianne; Gillotin, Florian; Somers, Fabian; Chiap, Patrice; Lebrun, Philippe; Pirotte, Bernard
Informations sur la publication:Journal of medicinal chemistry, 54, 24, page (8353-8361)
Statut de publication:Publié, 2011-12
Sujet CREF:Sciences bio-médicales et agricoles
Note générale:Journal Article
Research Support, Non-U.S. Gov't
SCOPUS: ar.j
Langue:Anglais
Identificateurs:urn:issn:0022-2623
info:doi/10.1021/jm200786z
info:scp/84055211840
info:pmid/22077416