Titre:
  • KATP channel openers: tissue selectivity of original 3-alkylaminopyrido- and 3-alkylaminobenzothiadiazine 1,1-dioxides.
Auteur:Lebrun, Philippe; Becker, Bénédicte; Morel, Nicole; Ghisdal, Philippe; Antoine, Marie-Hélène; de Tullio, Pascal; Pirotte, Bernard
Informations sur la publication:Biochemical pharmacology, 75, 2, page (468-475)
Statut de publication:Publié, 2008-01
Sujet CREF:Sciences bio-médicales et agricoles
Mots-clés:ATP-sensitive K+ channel
Benzothiadiazine dioxides
Insulin-secreting cell
KATP channel openers
Pyridothiadiazine dioxides
Vascular smooth muscle
MeSH keywords:Animals
Aorta -- drug effects
Aorta -- physiology
Glyburide -- pharmacology
Insulin -- secretion
KATP Channels -- drug effects
Membrane Potentials -- drug effects
Organ Specificity
Rats
Rats, Wistar
Structure-Activity Relationship
Thiadiazines -- pharmacology
Vasoconstriction -- drug effects
Note générale:In Vitro
Journal Article
Research Support, Non-U.S. Gov't
Langue:Anglais
Identificateurs:urn:issn:0006-2952
info:doi/10.1016/j.bcp.2007.08.032
info:pii/S0006-2952(07)00593-X
info:scp/37349016003
info:pmid/17920043