Titre:
  • Identification and pharmacological properties of E339-3D6, the first nonpeptidic apelin receptor agonist.
Auteur:Iturrioz, Xavier; Alvear-Perez, Rodrigo; De Mota, Nadia; Franchet, Christel; Guillier, Fabrice; Leroux, Vincent; Dabire, Hubert; Le Jouan, Melissande; Chabane, Hadjila; Gerbier, Romain; Bonnet, Dominique; Berdeaux, Alain; Maigret, Bernard; Galzi, Jean-Luc; Hibert, Marcel; Llorens-Cortes, Catherine
Informations sur la publication:The FASEB journal, 24, 5, page (1506-1517)
Statut de publication:Publié, 2010-05
Sujet CREF:Sciences bio-médicales et agricoles
Sciences exactes et naturelles
MeSH keywords:Animals
Aorta -- drug effects
Colforsin -- pharmacology
Cyclic AMP -- metabolism
Dipeptides -- chemistry -- isolation & purification -- pharmacology
Drug Evaluation, Preclinical -- methods
Fluoresceins -- chemistry -- isolation & purification -- pharmacology
Fluorescence Resonance Energy Transfer -- methods
Humans
Male
Mice
Rats
Rats, Inbred WKY
Receptors, G-Protein-Coupled -- agonists
Vasodilation
Vasopressins -- metabolism
Langue:Anglais
Identificateurs:urn:issn:0892-6638
info:doi/10.1096/fj.09-140715
info:pii/fj.09-140715
info:pmid/20040517